Ertugliflozin L-pyroglutamic acid
CAS No. 1210344-83-4
Ertugliflozin L-pyroglutamic acid ( PF-04971729 L-pyroglutamic acid )
Catalog No. M26680 CAS No. 1210344-83-4
Ertugliflozin L-pyroglutamic acid is a selective and orally active hSGLT2 inhibitor with an IC50 of 0.877 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
5MG | 35 | In Stock |
|
10MG | 50 | In Stock |
|
25MG | 74 | In Stock |
|
50MG | 87 | In Stock |
|
100MG | 129 | In Stock |
|
200MG | 188 | In Stock |
|
500MG | 322 | In Stock |
|
1G | Get Quote | In Stock |
|
Biological Information
-
Product NameErtugliflozin L-pyroglutamic acid
-
NoteResearch use only, not for human use.
-
Brief DescriptionErtugliflozin L-pyroglutamic acid is a selective and orally active hSGLT2 inhibitor with an IC50 of 0.877 nM.
-
DescriptionErtugliflozin L-pyroglutamic acid is a selective and orally active hSGLT2 inhibitor with an IC50 of 0.877 nM. Ertugliflozin L-pyroglutamic acid can be used for studies about the treatment of type 2 diabetes mellitus.(In Vitro):Ertugliflozin L-pyroglutamic acid demonstrated >2000-fold selectivity for SGLT2 over SGLT.(In Vivo):The oral administration of Ertugliflozin L-pyroglutamic to rats acid showed concentration-dependent glucosuria.
-
SynonymsPF-04971729 L-pyroglutamic acid
-
PathwayOthers
-
TargetOther Targets
-
RecptorCaspase-3
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number1210344-83-4
-
Formula Weight566.0
-
Molecular FormulaC27H32ClNO10
-
Purity>98% (HPLC)
-
Solubility——
-
SMILESOC(=O)[C@@H]1CCC(=O)N1.CCOc1ccc(Cc2cc(ccc2Cl)[C@]23OC[C@](CO)(O2)[C@@H](O)[C@H](O)[C@H]3O)cc1
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1.Kravchenko DV, et al. Synthesis and structure-activity relationship of 4-substituted 2-(2-acetyloxyethyl)-8-(morpholine-4-sulfonyl)pyrrolo[3,4-c]quinoline-1,3-diones as potent caspase-3 inhibitors. J Med Chem. 2005 Jun 2;48(11):3680-3.
molnova catalog
related products
-
1-Undecanol
1-Undecanol is a natural product in many foods such as fruits butter eggs and cooked pork is used as a flavoring ingredient.?
-
Exendin-4 peptide de...
FTSDVSKQMEEEAVRLFIEWLKNGGPSSGAPPPS is an Exendin-4 peptide derivative.Exendin-4 peptide derivatives are structurally derived from Exendin-4 and may relates to dual GLP-1/glucagon receptor agonists.
-
CCP peptide
CCP peptide is a synthetic cyclic peptide incorporating the amino acid citrulline.